Synthesis and Evaluation of Novel Inhibitors of Pim-1 and Pim-2 Protein Kinases-Reference-Cited by-同舟云学术

Synthesis and Evaluation of Novel Inhibitors of Pim-1 and Pim-2 Protein Kinases

Published:2008-12-15 Issue:1 Volume:52 Page:74-86
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Xia Zuping¹,Knaak Christian¹,Ma Jian¹,Beharry Zanna M.¹,McInnes Campbell¹,Wang Wenxue¹,Kraft Andrew S.¹,Smith Charles D.¹

Affiliation:

1. Department of Pharmaceutical and Biomedical Sciences, South Carolina College of Pharmacy, Medical University of South Carolina, 280 Calhoun Street, MSC140, Charleston, South Carolina, Department of Medicine, Medical University of South Carolina, Charleston, South Carolina, Department of Pharmaceutical and Biomedical Sciences, South Carolina College of Pharmacy, University of South Carolina, Columbia, South Carolina

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm800937p

Reference33 articles.

1. Proviral activation of the putative oncogene Pim-1 in MuLV induced T-cell lymphomas.

2. Delineation of prognostic biomarkers in prostate cancer

3. Pim-2 upregulation: Biological implications associated with disease progression and perinueral invasion in prostate cancer

4. Overexpression of PIM-1 is a potential biomarker in prostate carcinoma

5. Pim-1 expression in prostatic intraepithelial neoplasia and human prostate cancer

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