Identification of Novel Inhibitors of the Transforming Growth Factor β1 (TGF-β1) Type 1 Receptor (ALK5)-Reference-Cited by-同舟云学术

Identification of Novel Inhibitors of the Transforming Growth Factor β1 (TGF-β1) Type 1 Receptor (ALK5)

Published:2002-01-30 Issue:5 Volume:45 Page:999-1001
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Callahan James F.¹,Burgess Joelle L.¹,Fornwald James A.¹,Gaster Laramie M.¹,Harling John D.¹,Harrington Frank P.¹,Heer Jag¹,Kwon Chet¹,Lehr Ruth¹,Mathur A.¹,Olson Barbara A.¹,Weinstock Joseph¹,Laping Nicholas J.¹

Affiliation:

1. Department of Medicinal Chemistry, GlaxoSmithKline Pharmaceuticals, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426, Departments of Medicinal Chemistry, Renal Pharmacology, Protein Biochemistry, and Gene Expression Sciences, GlaxoSmithKline Pharmaceuticals, 709 Swedeland Road, King of Prussia, Pennsylvania 19406, and Department of Medicinal Chemistry, New Frontiers Science Park (North), Coldharbour Road, Harlow, Essex CM19 5AD, England

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm010493y

Reference17 articles.

1. TGF-β: Regulation of extracellular matrix

2. Production of extracellular matrix by glomerular epithelial cells is regulated by transforming growth factor-β1

3. Effects of transforming growth factor-?1 on the extracellular matrix and cytoskeleton of cultured astrocytes

4. How cells read TGF-β signals

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