Virtual Screening and X-ray Crystallography for Human Kallikrein 6 Inhibitors with an Amidinothiophene P1 Group-Reference-Cited by-同舟云学术

Virtual Screening and X-ray Crystallography for Human Kallikrein 6 Inhibitors with an Amidinothiophene P1 Group

Published:2012-01-17 Issue:2 Volume:3 Page:159-164
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Liang Guyan¹,Chen Xin¹,Aldous Suzanne¹,Pu Su-Fen¹,Mehdi Shujaath¹,Powers Elaine¹,Giovanni Andrew¹,Kongsamut Sathapana¹,Xia Tianhui¹,Zhang Ying¹,Wang Rachel¹,Gao Zhongli¹,Merriman Gregory¹,McLean Larry R.¹,Morize Isabelle¹

Affiliation:

1. Molecular Innovative Therapeutics, ‡Fibrosis and Wound Repair, §Global Pharmacovigilance & Epidemiology, ∥Immunology and Inflammation Unit, ⊥Early to Candidate Unit, #Aging Therapeutic Unit, and ∇Biologics, Sanofi Pharmaceuticals, 1041 Route 202/206, Mailstop 203A, Bridgewater, New Jersey 08807, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml200291e

Reference31 articles.

1. A comprehensive nomenclature for serine proteases with homology to tissue kallikreins

2. Kallikrein-related peptidases

3. Managing Peptidases in the Genomic Era

4. Chao, J.Human kallikrein 1, tissue kallikrein.Handbook of Proteolytic Enzymes,2nd ed.Elsevier Academic Press:Amsterdam, Boston, 2004; Vol.2, p1577.

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