DNA Methylation Bisubstrate Inhibitors Are Fast-Acting Drugs Active against Artemisinin-Resistant Plasmodium falciparum Parasites-Reference-Cited by-同舟云学术

DNA Methylation Bisubstrate Inhibitors Are Fast-Acting Drugs Active against Artemisinin-Resistant Plasmodium falciparum Parasites

Published:2019-11-27 Issue:1 Volume:6 Page:16-21
ISSN:2374-7943
Container-title:ACS Central Science
language:en
Short-container-title:ACS Cent. Sci.

Author:

Nardella Flore¹,Halby Ludovic²,Hammam Elie¹³,Erdmann Diane²⁴,Cadet-Daniel Véronique²,Peronet Roger¹,Ménard Didier¹⁵,Witkowski Benoit⁵,Mecheri Salah¹,Scherf Artur¹,Arimondo Paola B.²^ORCID

Affiliation:

1. Unité Biologie des Interactions Hôte-Parasite, Département de Parasites et Insectes Vecteurs, Institut Pasteur, CNRS ERL 9195, INSERM Unit U1201, 25-28 Rue du Dr Roux, Paris 75015, France

2. Epigenetic Chemical Biology, Department of Structural Biology and Chemistry, Institut Pasteur, UMR n°3523, CNRS, 28 Rue du Dr Roux, Paris 75015, France

3. Ecole Doctorale Complexité du Vivant ED515, Sorbonne Universités, Paris 6, Paris 75005, France

4. Ecole Doctorale MTCI ED563, Université de Paris, Sorbonne Paris Cité, Paris 75006, France

5. Malaria Molecular Epidemiology Unit, Pasteur Institute in Cambodia, Phnom Penh, Cambodia

Funder

DIM1 Health Ile de France 2019

DARRI Carnot Pasteur MS 2019

French Parasitology consortium ParaFrap

Fondation Pasteur Swiss grant

PTR Institut Pasteur 2019

ERC Advanced grant

Publisher

American Chemical Society (ACS)

Subject

General Chemical Engineering,General Chemistry

Link

http://pubs.acs.org/doi/pdf/10.1021/acscentsci.9b00874

Reference26 articles.

1. World Health Organization. World malaria report; World Health Organization, 2018; pp xii–xiii, https://www.who.int/malaria/publications/world-malaria-report-2018/report/en/.

2. Malaria Epigenetics

3. Antigenic Variation in Plasmodium falciparum

4. Post-translational protein modifications in malaria parasites

5. Small-molecule histone methyltransferase inhibitors display rapid antimalarial activity against all blood stage forms in Plasmodium falciparum

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