Allosteric Modulators Enhancing GLP-1 Binding to GLP-1R via a Transmembrane Site

Author:

Wang Jiang123,Yang Dehua1,Cheng Xi13,Yang Linlin4,Wang Zhaohui1,Dai Antao1,Cai Xiaoqing1,Zhang Chao5,Yuliantie Elita1,Liu Qiaofeng6,Jiang Hualiang123,Liu Hong123ORCID,Wang Ming-Wei127,Yang Huaiyu8ORCID

Affiliation:

1. State Key Laboratory of Drug Research, The National Center for Drug Screening and CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China

2. University of Chinese Academy of Sciences, Beijing 100049, China

3. School of Pharmaceutical Science and Technology, Hangzhou Institute of Advanced Study, Hangzhou 310024, China

4. Department of Pharmacology, School of Basic Medical Sciences, Zhengzhou University, Zhengzhou 450001, China

5. School of Life Science and Technology, ShanghaiTech University, Shanghai 201210, China

6. School of Pharmacy, Fudan University, Shanghai 201203, China

7. Department of Pharmacology, School of Basic Medical Sciences, Fudan University, Shanghai 200032, China

8. Shanghai Key Laboratory of Regulatory Biology, Institute of Biomedical Sciences, School of Life Sciences, East China Normal University, Shanghai 200241, China

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

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