Molecular Mechanisms of Desensitization Underlying the Differential Effects of Formyl Peptide Receptor 2 Agonists on Cardiac Structure–Function Post Myocardial Infarction

Author:

Lupisella John1ORCID,St-Onge Stéphane2,Carrier Marilyn2,Cook Erica M.3,Wang Tao3,Sum Chi3,Fernando Gayani1,Apgar Kendra1,Zhang Rongan1,Carson Nancy1,Snyder Bradley J.1,Ryan Carol S.1,Ma Xiuying1,Dierks Elizabeth A.4,Little Sean1,Kick Ellen K.5ORCID,Wurtz Nicholas R.5ORCID,Bouvier Michel2ORCID,Héroux Madeleine2,Garcia Ricardo A.1

Affiliation:

1. Department of Cardiovascular and Fibrosis Drug Discovery, Bristol Myers Squibb, P.O. Box 4000 Princeton, New Jersey08543-4000, United States

2. Institute for Research in Immunology and Cancer, Université de Montréal, QuebecH3T 1J4, Canada

3. Department of Lead Discovery and Optimization, Bristol Myers Squibb, P.O. Box 4000 Princeton, New Jersey08543-4000, United States

4. Department of Drug Metabolism and Pharmacokinetics, Bristol Myers Squibb, P.O. Box 4000 Princeton, New Jersey08543-4000, United States

5. Department of Cardiovascular Discovery Chemistry, Bristol Myers Squibb, P.O. Box 4000 Princeton, New Jersey08543-4000, United States

Publisher

American Chemical Society (ACS)

Subject

Pharmacology (medical),Pharmacology

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