Pyrazolones Potentiate Colistin Activity against MCR-1-Producing Resistant Bacteria: Computational and Microbiological Study

Author:

Hanpaibool Chonnikan1,Ngamwongsatit Natharin23ORCID,Ounjai Puey45ORCID,Yotphan Sirilata6,Wolschann Peter7,Mulholland Adrian J.8ORCID,Spencer James9ORCID,Rungrotmongkol Thanyada110

Affiliation:

1. Center of Excellence in Biocatalyst and Sustainable Biotechnology, Department of Biochemistry, Faculty of Science, Chulalongkorn University, Bangkok 10330, Thailand

2. Department of Clinical Sciences and Public Health, Faculty of Veterinary Science, Mahidol University, Nakhon Pathom 73170, Thailand

3. Laboratory of Bacteria, Veterinary Diagnostic Center, Faculty of Veterinary Science, Mahidol University, Nakhon Pathom 73170, Thailand

4. Department of Biology, Faculty of Science, Mahidol University, Bangkok 10400, Thailand

5. Center of Excellence on Environmental Health and Toxicology, Office of Higher Education Commission, Ministry of Education, Bangkok 10400, Thailand

6. Center of Excellence for Innovation in Chemistry (PERCH-CIC), Department of Chemistry, Faculty of Science, Mahidol University, Bangkok 10400, Thailand

7. Institute of Theoretical Chemistry, University of Vienna, Vienna 1090, Austria

8. Centre for Computational Chemistry, School of Chemistry, University of Bristol, Bristol BS8 1TS, U.K.

9. School of Cellular and Molecular Medicine, University of Bristol, Bristol BS8 1TD, U.K.

10. Program in Bioinformatics and Computational Biology, Graduate School, Chulalongkorn University, Bangkok 10400, Thailand

Funder

Engineering and Physical Sciences Research Council

Medical Research Council

Chulalongkorn University

Publisher

American Chemical Society (ACS)

Subject

General Chemical Engineering,General Chemistry

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