Structure-Based Discovery of A2A Adenosine Receptor Ligands-Reference-Cited by-同舟云学术

Structure-Based Discovery of A2A Adenosine Receptor Ligands

Published:2010-04-20 Issue:9 Volume:53 Page:3748-3755
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Carlsson Jens¹,Yoo Lena²,Gao Zhan-Guo²,Irwin John J.¹,Shoichet Brian K.¹,Jacobson Kenneth A.²

Affiliation:

1. Department of Pharmaceutical Chemistry, University of California, 1700 4th Street, Box 2550, San Francisco, California 94158

2. Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, National Institutes of Health, Bethesda, Maryland 20892

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm100240h

Reference56 articles.

1. How many drug targets are there?

2. High-Resolution Crystal Structure of an Engineered Human β 2 -Adrenergic G Protein–Coupled Receptor

3. GPCR Engineering Yields High-Resolution Structural Insights into β 2 -Adrenergic Receptor Function

4. Structure of a β1-adrenergic G-protein-coupled receptor

5. The 2.6 Angstrom Crystal Structure of a Human A 2A Adenosine Receptor Bound to an Antagonist

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