A Method for Identifying and Developing Functional Group Tolerant Catalytic Reactions: Application to the Buchwald–Hartwig Amination-Reference-Cited by-同舟云学术

A Method for Identifying and Developing Functional Group Tolerant Catalytic Reactions: Application to the Buchwald–Hartwig Amination

Published:2017-03-15 Issue:7 Volume:82 Page:3741-3750
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Richardson Jeffery¹^ORCID,Ruble J. Craig²,Love Elizabeth A.³,Berritt Simon⁴

Affiliation:

1. Discovery Chemistry Research and Technologies, Eli Lilly and Company Limited, Erl Wood Manor, Windlesham, Surrey GU20 6PH, United Kingdom

2. Discovery Chemistry Research and Technologies, Eli Lilly and Company, Indianapolis, Indiana 46285, United States

3. Translational Research Office Drug Discovery Group, University College London School of Pharmacy, 29−39 Brunswick Square, London WC1N 1AX, United Kingdom

4. Penn/Merck Laboratory for High-Throughput Experimentation, Department of Chemistry, University of Pennsylvania, 231 South 34th Street, Philadelphia, Pennsylvania 19104-6323, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.joc.7b00201

Reference48 articles.

1. Nanomole-scale high-throughput chemistry for the synthesis of complex molecules

2. Factors Determining the Selection of Organic Reactions by Medicinal Chemists and the Use of These Reactions in Arrays (Small Focused Libraries)

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4. Finding the sweet spot: the role of nature and nurture in medicinal chemistry

5. Big Data from Pharmaceutical Patents: A Computational Analysis of Medicinal Chemists’ Bread and Butter

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