Umpolung Flow Chemistry for the Synthesis of a 3-Oxo-3H-spiro[benzofuran-2,4′-piperidine] Building Block

Author:

Pompeo Matthew M.1ORCID,Kelly Sean M.1ORCID,St-Jean Frédéric1ORCID,Bass Thomas M.1,Dalton Derek M.1ORCID,Zell Daniel1ORCID,Han Chong1ORCID,Sirois Lauren E.1ORCID,Gosselin Francis1ORCID

Affiliation:

1. Department of Synthetic Molecule Process Chemistry, Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States

Publisher

American Chemical Society (ACS)

Reference32 articles.

1. Identification of GDC-1971 (RLY-1971), a SHP2 Inhibitor Designed for the Treatment of Solid Tumors

2. Recent Advances of SHP2 Inhibitors in Cancer Therapy: Current Development and Clinical Application

3. a Study to Evaluate the Safety, Pharmacokinetics, and Activity of GDC-1971 in Combination With Either Osimertinib in Participants With Unresectable, Locally Advanced, or Metastatic Non-Small Cell Lung Cancer, or With Cetuximab in Participants With Metastatic Colorectal Cancer, NCT05954871, 2023.

4. bF. Hoffmann-La Roche Ltd A Study to Evaluate the Safety, Pharmacokinetics, and Activity of GDC-1971 in Combination With Atezolizumab in Participants With Locally Advanced or Metastatic Solid Tumors, NCT05487235, 2022.

5. c A Phase Ia/Ib Dose-Escalation and Dose-Expansion Study Evaluating the Safety, Pharmacokinetics, and Activity of GDC-6036 as a Single Agent and in Combination With Other Anti-cancer Therapies in Patients With Advanced or Metastatic Solid Tumors With a KRAS G12C Mutation, NCT04449874, 2020.

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