Selective Non-nucleoside Inhibitors of Human DNA Methyltransferases Active in Cancer Including in Cancer Stem Cells

Author:

Valente Sergio1,Liu Yiwei2,Schnekenburger Michael3,Zwergel Clemens14,Cosconati Sandro5,Gros Christina6,Tardugno Maria1,Labella Donatella1,Florean Cristina3,Minden Steven3,Hashimoto Hideharu2,Chang Yanqi2,Zhang Xing2,Kirsch Gilbert4,Novellino Ettore7,Arimondo Paola B.6,Miele Evelina8,Ferretti Elisabetta9,Gulino Alberto9,Diederich Marc310,Cheng Xiaodong2,Mai Antonello1

Affiliation:

1. Dipartimento di Chimica e Tecnologie del Farmaco, Sapienza Università di Roma, P.le Aldo Moro 5, 00185 Roma, Italy

2. Department of Biochemistry, Emory University School of Medicine, 1510 Clifton Road, Atlanta, Georgia 30322, United States

3. Laboratoire de Biologie Moléculaire et Cellulaire du Cancer (LBMCC), Hôpital Kirchberg, 9, rue Edward Steichen, L-2540 Luxembourg

4. Laboratoire d’Ingénierie Moléculaire et Biochimie Pharmacologique, Université de Lorraine−Metz, 1 Boulevard Arago, 57070 Metz, France

5. DiSTABiF, Seconda Università di Napoli, Via G. Vivaldi 43, 81100 Caserta, Italy

6. USR3388 CNRS-Pierre Fabre ETaC, CRDPF, 3 Avenue H. Curien, 31035 Toulouse Cedex 01, France

7. Dipartimento di Farmacia, Università di Napoli “Federico II”, Via D. Montesano, 49, 80131 Napoli, Italy

8. Istituto Italiano di Tecnologia and Dipartimento of Medicina Molecolare, Sapienza Università di Roma, Viale Regina Elena 291, 00161 Roma, Italy

9. Dipartimento di Medicina Sperimentale e Dipartimento di Medicina Molecolare, Sapienza Università di Roma, Viale Regina Elena 291, 00161 Rome, Italy

10. Department of Pharmacy, College of Pharmacy, Seoul National University, 599 Gwanak-ro, Gwanak-gu, Seoul 151-742, Korea

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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