A New-Class Antibacterial—Almost. Lessons in Drug Discovery and Development: A Critical Analysis of More than 50 Years of Effort toward ATPase Inhibitors of DNA Gyrase and Topoisomerase IV
Author:
Affiliation:
1. AstraZeneca, 35 Gatehouse Drive, Waltham, Massachusetts 02451, United States
Publisher
American Chemical Society (ACS)
Subject
Infectious Diseases
Link
https://pubs.acs.org/doi/pdf/10.1021/id500013t
Reference234 articles.
1. Bryskier, A.InAntibiotics and Antibacterial Agents: Classifications and Structure-Activity Relationship;Bryskier, A., Ed.; Antimicrobial agents: antibacterials and antifungals;ASM Press:Washington, DC, 2005; pp13–38.
2. Antibacterial discovery and development—the failure of success?
3. Challenges of antibacterial discovery revisited
4. The 10 × ‘20 Initiative: Pursuing a Global Commitment to Develop 10 New Antibacterial Drugs by 2020
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