Cyclic Peptides KS-133 and KS-487 Multifunctionalized Nanoparticles Enable Efficient Brain Targeting for Treating Schizophrenia

Author:

Sakamoto Kotaro1,Iwata Seigo2,Jin Zihao34,Chen Lu3,Miyaoka Tatsunori3ORCID,Yamada Mei3,Katahira Kaiga3,Yokoyama Rei45,Ono Ami46,Asano Satoshi4,Tanimoto Kotaro6,Ishimura Rika7,Nakagawa Shinsaku378,Hirokawa Takatsugu910ORCID,Ago Yukio348,Miyako Eijiro2ORCID

Affiliation:

1. Research & Development Department, Ichimaru Pharcos Company Limited, 318-1 Asagi, Motosu, 501-0475 Gifu, Japan

2. Graduate School of Advanced Science and Technology, Japan Advanced Institute of Science and Technology, 1-1 Asahidai, Nomi, 923-1292 Ishikawa, Japan

3. Laboratory of Biopharmaceutics, Osaka University, 1-6 Yamada-oka, Suita, 565-0871 Osaka, Japan

4. Department of Cellular and Molecular Pharmacology, Graduate School of Biomedical and Health Sciences, Hiroshima University, 1-2-3 Kasumi, Minami-ku, Hiroshima, 734-8553 Hiroshima, Japan

5. Laboratory of Molecular Neuropharmacology, Osaka University, 1-6 Yamada-oka, Suita, 565-0871 Osaka, Japan

6. Department of Orthodontics and Craniofacial Developmental Biology, Graduate School of Biomedical and Health Sciences, Hiroshima University, 1-2-3 Kasumi, Minami-ku, Hiroshima, 734-8553 Hiroshima, Japan

7. Center for Supporting Drug Discovery and Life Science Research, Graduate School of Pharmaceutical Science, Osaka University, 1-6 Yamada-oka, Suita, 565-0871 Osaka, Japan

8. Global Center for Medical Engineering and Informatics, Osaka University, 2-2 Yamada-oka, Suita, 565-0871 Osaka Japan

9. Division of Biomedical Science, Institute of Medicine, University of Tsukuba, 1-1-1 Tennodai, 305-8575 Tsukuba, Japan

10. Transborder Medical Research Center, University of Tsukuba, 1-1-1 Tennodai, 305-8575 Tsukuba, Japan

Funder

Institute for Fermentation, Osaka

Japan Agency for Medical Research and Development

Adaptable and Seamless Technology Transfer Program through Target-Driven R and D

Tokyo Biochemical Research Foundation

Japan Society for the Promotion of Science

Japan Science and Technology Agency

Uehara Memorial Foundation

Publisher

American Chemical Society (ACS)

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