Serotonin 5-HT2 Receptor, Dopamine D2 Receptor, and α1 Adrenoceptor Antagonists. Conformationally Flexible Analogues of the Atypical Antipsychotic Sertindole-Reference-Cited by-同舟云学术

Serotonin 5-HT2 Receptor, Dopamine D2 Receptor, and α1 Adrenoceptor Antagonists. Conformationally Flexible Analogues of the Atypical Antipsychotic Sertindole

Published:1996-01-01 Issue:19 Volume:39 Page:3723-3738
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Andersen Kim¹,Liljefors Tommy¹,Hyttel John¹,Perregaard Jens¹

Affiliation:

1. Research Departments, H. Lundbeck A/S, Ottiliavej 9, DK-2500 Copenhagen, Denmark, and Department of Medicinal Chemistry, Royal Danish School of Pharmacy Universitetsparken, DK-2100 Copenhagen Ø, Denmark

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm960159f

Reference52 articles.

1. Sertindole, a new neuroleptic with extreme selectivity on A10 versus A9 dopamine neurones in the rat

2. Electrophysiological profile of the new atypical neuroleptic, sertindole, on midbrain dopamine neurones in rats: Acute and repeated treatment

3. Neurochemical and in vivo pharmacological profile of sertindole, a limbic-selective neuroleptic compound

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