On the Origin of the Different Reversible Characters of Salinosporamide A and Homosalinosporamide A in the Covalent Inhibition of the Human 20S Proteasome
Author:
Affiliation:
1. Biocomp Group, Institute of Advanced Materials (INAM), Universitat Jaume I, 12071 Castellón, Spain
Funder
Generalitat Valenciana
Universitat Jaume I
Ministerio de Ciencia e Innovaci??n
Ministerio de Econom??a y Competitividad
Publisher
American Chemical Society (ACS)
Subject
Catalysis,General Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acscatal.1c02614
Reference100 articles.
1. A Perspective on the Kinetics of Covalent and Irreversible Inhibition
2. Structure of Mpro from SARS-CoV-2 and discovery of its inhibitors
3. Many small steps towards a COVID-19 drug
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5. Discovery of Ketone-Based Covalent Inhibitors of Coronavirus 3CL Proteases for the Potential Therapeutic Treatment of COVID-19
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