2-Azidobenzaldehyde-Based [4+2] Annulation for the Synthesis of Quinoline Derivatives-Reference-Cited by-同舟云学术

2-Azidobenzaldehyde-Based [4+2] Annulation for the Synthesis of Quinoline Derivatives

Published:2024-03-11 Issue:6 Volume:29 Page:1241
ISSN:1420-3049
Container-title:Molecules
language:en
Short-container-title:Molecules

Author:

Zhang Xiaofeng¹²,Liu Miao¹³,Qiu Weiqi¹⁴,Zhang Wei¹^ORCID

Affiliation:

1. Center for Green Chemistry and Department of Chemistry, University of Massachusetts Boston, 100 Morrissey Blvd, Boston, MA 02125, USA

2. Department of Medicinal Chemistry, Cerevel Therapeutics, Cambridge, MA 02141, USA

3. Department of Mechanical Engineering, University of Wisconsin Milwaukee, Milwaukee, WI 53211, USA

4. Department of Chemistry, Boston College, 2609 Beacon Street, Chestnut Hill, MA 20467, USA

Abstract

Quinoline is a privileged heterocyclic ring which can be found in many drug molecules and bioactive compounds. The development of synthetic methods for making quinoline derivatives continuously attracts the interest of organic and medicinal chemists. This paper highlights 2-azidobenzaldehyde-based [4+2] annulation for the synthesis of quinoline derivatives including fused and spiro-quinolines, quinoline-4-ols, 4-aminoquinolines, and related compounds.

Publisher

MDPI AG

Link

https://www.mdpi.com/1420-3049/29/6/1241/pdf

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