Inhibition of Autophagy by a Small Molecule through Covalent Modification of the LC3 Protein

Author:

Fan Shijie12,Yue Liyan1,Wan Wei12,Zhang Yuanyuan12,Zhang Bidong1,Otomo Chinatsu3,Li Quanfu4,Lin Tingting15,Hu Junchi6,Xu Pan1,Zhu Mingrui1,Tao Hongru1,Chen Zhifeng1,Li Lianchun1,Ding Hong1,Yao Zhiyi7,Lu Junyan1,Wen Yi1,Zhang Naixia1,Tan Minjia1,Chen Kaixian12,Xie Yuli7,Otomo Takanori3,Zhou Bing8,Jiang Hualiang12,Dang Yongjun46,Luo Cheng125910ORCID

Affiliation:

1. The Center for Chemical Biology, Drug Discovery and Design Center State Key Laboratory of Drug Research Shanghai Institute of Materia Medica Chinese Academy of Sciences Shanghai 201203 China

2. University of Chinese Academy of Sciences No.19A Yuquan Road Beijing 100049 China

3. Department of Integrative Structural and Computational Biology The Scripps Research Institute La Jolla CA 92037 USA

4. Key Laboratory of Metabolism and Molecular Medicine the Ministry of Education Department of Biochemistry and Molecular Biology School of Basic Medical Sciences Fudan University Shanghai 200032 China

5. School of Life Science and Technology ShanghaiTech University 100 Haike Road Shanghai 201210 China

6. Center for Novel Target and Therapeutic Intervention Institute of Life Sciences Chongqing Medical University No. 1, Yixueyuan Road, Yuzhong District Chongqing China

7. Suzhou Autopharm 108 Yuxin Road Jiangsu 215123 China

8. Department of Medicinal Chemistry State Key Laboratory of Drug Research Shanghai Institute of Materia Medica Chinese Academy of Sciences 555 Zuchongzhi Road Shanghai 201203 China

9. School of Pharmacy Fudan University Shanghai 201203 China

10. School of Pharmaceutical Sciences Zhejiang Chinese Medical University Hangzhou 310053 China

Funder

National Natural Science Foundation of China

Science and Technology Commission of Shanghai Municipality

Foundation for the National Institutes of Health

Publisher

Wiley

Subject

General Chemistry,Catalysis

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