Repurposing the selective estrogen receptor modulator bazedoxifene to suppress gastrointestinal cancer growth

Author:

Thilakasiri Pathum1,Huynh Jennifer1,Poh Ashleigh R1,Tan Chin Wee2,Nero Tracy L34,Tran Kelly1,Parslow Adam C15,Afshar‐Sterle Shoukat1,Baloyan David1,Hannan Natalie J6,Buchert Michael1,Scott Andrew Mark157,Griffin Michael DW4,Hollande Frederic8,Parker Michael W34,Putoczki Tracy L2,Ernst Matthias1ORCID,Chand Ashwini L1ORCID

Affiliation:

1. Olivia Newton‐John Cancer Research Institute School of Cancer Medicine La Trobe University Heidelberg Vic. Australia

2. The Walter and Eliza Hall Institute Melbourne Vic. Australia

3. ACRF Rational Drug Discovery Centre St Vincent's Institute Melbourne Vic. Australia

4. Department of Biochemistry and Molecular Biology Bio21 Institute University of Melbourne Melbourne Vic. Australia

5. Department of Molecular Imaging and Therapy Austin Health Melbourne Vic. Australia

6. Department of Obstetrics and Gynaecology University of Melbourne Melbourne Vic. Australia

7. Department of Medicine University of Melbourne Melbourne Vic. Australia

8. Department of Clinical Pathology University of Melbourne Centre for Cancer Research Victorian Comprehensive Cancer Centre University of Melbourne Melbourne Vic. Australia

Funder

National Health and Medical Research Council

Australian Research Council

Cancer Australia

Ludwig Institute for Cancer Research

Cure Brain Cancer Foundation

Cancer Council Victoria

Publisher

EMBO

Subject

Molecular Medicine

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