Carfilzomib induces leukaemia cell apoptosis via inhibiting ELK1/KIAA1524 (Elk-1/CIP2A) and activating PP2A not related to proteasome inhibition

Author:

Liu Chun-Yu1234,Hsieh Feng-Shu5,Chu Pei-Yi67,Tsai Wen-Chun2,Huang Chun-Teng38,Yu Yuan-Bin34,Huang Tzu-Ting12,Ko Po-Shen234,Hung Man-Hsin234,Wang Wan-Lun2,Shiau Chung-Wai9,Chen Kuen-Feng510ORCID

Affiliation:

1. Comprehensive Breast Health Centre; Taipei Veterans General Hospital; Taipei Taiwan

2. Division of Medical Oncology; Department of Oncology; Taipei Veterans General Hospital; Taipei Taiwan

3. School of Medicine; National Yang-Ming University; Taipei Taiwan

4. Division of Haematology and Oncology; Department of Medicine; Taipei Veterans General Hospital; Taipei Taiwan

5. Department of Medical Research; National Taiwan University Hospital; Taipei Taiwan

6. Department of Pathology; Show Chwan Memorial Hospital; Changhua Taiwan

7. School of Medicine; Fu Jen Catholic University; New Taipei City Taiwan

8. Division of Haematology and Oncology; Department of Medicine; Yang-Ming Branch of Taipei City Hospital; Taipei Taiwan

9. Institute of Biopharmaceutical Sciences; National Yang-Ming University; Taipei Taiwan

10. National Center of Excellence for Clinical Trial and Research; National Taiwan University Hospital; Taipei Taiwan

Funder

Yen Tjing Ling Medical Foundation

Ministry of Science and Technology, Taiwan

Yang-Ming Branch of Taipei City Hospital

Taipei Veterans General Hospital

TVGH-NTUH Joint Research Program

National Taiwan University Hospital

Chong Hin Loon Memorial Cancer

Biotherapy Research Centre of National Yang-Ming University, Taipei, Taiwan

Publisher

Wiley

Subject

Hematology

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