Solid-Supported Synthesis and 5-HT7/5-HT1AReceptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1H)-one-Reference-Cited by-同舟云学术

Solid-Supported Synthesis and 5-HT7/5-HT1AReceptor Affinity of Arylpiperazinylbutyl Derivatives of 4,5-dihydro-1,2,4-triazine-6-(1H)-one

Published:2015-03-06 Issue:4 Volume:86 Page:697-703
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Grychowska Katarzyna¹,Masurier Nicolas²,Verdié Pascal²,Satała Grzegorz³,Bojarski Andrzej J.³,Martinez Jean²,Pawłowski Maciej¹,Subra Gilles²,Zajdel Paweł¹

Affiliation:

1. Department of Medicinal Chemistry; Jagiellonian University Medical College; 9 Medyczna Street 30-688 Kraków Poland

2. Department of Aminoacids; Peptides and Proteins Institute of Biomolecules Max Mousseron; UMR CNRS 5247; 15 Charles Flahault Av. 34093 Montpellier France

3. Department of Medicinal Chemistry; Institute of Pharmacology; Polish Academy of Sciences; 12 Smętna Street 31-343 Kraków Poland

Funder

Polish Ministry of Science and Higher Education (MNiSW)

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/cbdd.12539/fullpdf

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5. (Phenylpiperazinyl-butyl)oxindoles as selective 5-HT7 receptor antagonists;Volk;J Med Chem,2008

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