Discovery of novel bacterial FabH inhibitors (Pyrazol-Benzimidazole amide derivatives): Design, synthesis, bioassay, molecular docking and crystal structure determination-Reference-Cited by-同舟云学术

Discovery of novel bacterial FabH inhibitors (Pyrazol-Benzimidazole amide derivatives): Design, synthesis, bioassay, molecular docking and crystal structure determination

Published:2019-06 Issue: Volume:171 Page:209-220
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Wang Yan-Ting,Shi Tian-Qi,Fu Jie^ORCID,Zhu Hai-Liang^ORCID

Funder

National Key R&D Program of China

China Postdoctoral Science Foundation

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference34 articles.

1. Designer antibacterial peptides kill fluoroquinolone-resistant clinical isolates;Otvos;J. Med. Chem.,2005

2. Design, synthesis and biological evaluation of urea derivatives from -hydroxybenzylamines and phenylisocyanate as potential FabH inhibitors;Li;Bioorg. Med. Chem.,2011

3. Syntheses and antibacterial activity of a series of 3-(pyridine-3-yl)-2-oxazolidinone;Cui;Eur. J. Med. Chem.,2005

4. Antimicrobial natural products as beta-ketoacyl-acyl carrier protein synthase III inhibitors;Lee;Bioorg. Med. Chem.,2009

5. Advances in the research of β-ketoacyl-ACP synthase III (FabH) inhibitors;HJ;Curr. Med. Chem.,2009

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