Discovery of novel non-steroidal selective glucocorticoid receptor modulators by structure- and IGN-based virtual screening, structural optimization, and biological evaluation

Author:

Hu Xueping,Pang Jinping,Chen Changwei,Jiang Dejun,Shen Chao,Chai Xin,Yang LiuORCID,Zhang Xujun,Xu Lei,Cui Sunliang,Hou Tingjun,Li DanORCID

Funder

National Natural Science Foundation of China

National Key Research and Development Program of China

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

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3. Benefits and harm of systemic steroids for short- and long-term use in rhinitis and rhinosinusitis: an Eaaci position paper;Hox;Clin. Transl. Allergy,2020

4. Eular recommendations for the management of rheumatoid arthritis with synthetic and biological disease-modifying antirheumatic drugs: 2019 update;Smolen;Ann. Rheum. Dis.,2020

5. Glucocorticoids, cytokines and brain abnormalities in depression;Zunszain;Prog. Neuro Psychopharmacol.,2011

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