Design, synthesis and biological evaluation of quinoxaline compounds as anti-HIV agents targeting reverse transcriptase enzyme

Author:

Fabian Lucas,Taverna Porro Marisa,Gómez Natalia,Salvatori Melina,Turk Gabriela,Estrin Darío,Moglioni AlbertinaORCID

Funder

Agencia Nacional de Promoción Científica y Tecnológica

Universidad de Buenos Aires

Consejo Nacional de Investigaciones Científicas y Técnicas

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference35 articles.

1. Emerging antiretroviral drugs;Fernández-Montero;Expert Opin. Pharmacother.,2014

2. Non-nucleoside reverse transcriptase inhibitors: a review on pharmacokinetics, pharmacodynamics, safety and tolerability;Usach;J. Int. AIDS Soc.,2013

3. Quinoxalinone as a privileged platform in drug development;Shi;Mini Rev. Med. Chem.,2018

4. Recent advances in pharmacological activities of quinoxaline derivatives;Husain;J. Pharm. Res.,2011

5. Preclinical evaluation of HBY 097, a new nonnucleoside reverse transcriptase inhibitor of human immunodeficiency virus type 1 replication;Kleim;J. Antimicrob. Chemother.,1995

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