Design, synthesis and antitrypanosomal activities of 2,6-disubstituted-4,5,7-trifluorobenzothiophenes-Reference-Cited by-同舟云学术

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Design, synthesis and antitrypanosomal activities of 2,6-disubstituted-4,5,7-trifluorobenzothiophenes

Published:2016-01 Issue: Volume:108 Page:347-353
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Bhambra Avninder S.,Edgar Mark,Elsegood Mark R.J.,Li Yuqi,Weaver George W.,Arroo Randolph R.J.,Yardley Vanessa,Burrell-Saward Hollie,Krystof Vladimir

Funder

Ministry of Education, Youth and Sports of the Czech Republic

Loughborough University

De Montfort University

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference29 articles.

1. Determination of an optimal dosing regimen for fexinidazole, a novel oral drug for the treatment of Human African Trypanosomiasis: first-in-human studies;Tarral;Clin. Pharmacokinet.,2014

2. 3-Nitrotriazole-based piperazides as potent antitrypanosomal agents;Papadopoulou;Eur. J. Med. Chem.,2015

3. Structure-activity relationship of hybrids of cinchona alkaloids and bile acids with in vitro antiplasmodial and antitrypanosomal activities;Leverrier;Eur. J. Med. Chem.,2015

4. Scaffold-based Drug Discovery in Structure-based Drug Discovery;Zhang,2007

5. Tetrahydropyrido[3,4-b]pyrazine scaffolds from pentafluoropyridine;Sandford;J. Org. Chem.,2005

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