Overview of human 20 alpha-hydroxysteroid dehydrogenase (AKR1C1): Functions, regulation, and structural insights of inhibitors

Author:

Chu Xianglin,He Siyu,Liu Yang,Liu Yijun,Feng Feng,Guo Qinglong,Zhao Li,Sun HaopengORCID

Funder

National Natural Science Foundation of China

Publisher

Elsevier BV

Subject

Toxicology,General Medicine

Reference215 articles.

1. The aldo-keto reductases (AKRs): Overview;Penning;Chem. Biol. Interact.,2015

2. Introduction and overview of the aldo-keto reductase superfamily;Penning;Abstr. Pap. Am. Chem. Soc.,2002

3. Promiscuity and diversity in 3-ketosteroid reductases;Penning;J. Steroid Biochem. Mol. Biol.,2015

4. Overview of AKR1C3: inhibitor achievements and disease insights;Liu;J. Med. Chem.,2020

5. Role of aldo-keto reductase family 1 (AKR1) enzymes in human steroid metabolism;Rizner;Steroids,2014

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