Potent and reversible open-channel blocker of NMDA receptor derived from dizocilpine with enhanced membrane-to-channel inhibition

Author:

Misiachna AnnaORCID,Konecny JanORCID,Kolcheva Marharyta,Ladislav MarekORCID,Prchal LukasORCID,Netolicky JakubORCID,Kortus StepanORCID,Zahumenska PetraORCID,Langore EmilyORCID,Novak Martin,Hemelikova KatarinaORCID,Hermanova ZuzanaORCID,Hrochova MichaelaORCID,Pelikanova AnezkaORCID,Odvarkova Jitka,Pejchal Jaroslav,Kassa Jiri,Zdarova Karasova Jana,Korabecny JanORCID,Soukup OndrejORCID,Horak Martin

Funder

MEYS CR

Publisher

Elsevier BV

Reference53 articles.

1. Antihistamine agent dimebon as a novel neuroprotector and a cognition enhancer;Bachurin;Ann. N. Y Acad. Sci.,2001

2. Nmda receptor affinities of 1,2-diphenylethylamine and 1-(1,2-diphenylethyl)piperidine enantiomers and of related compounds;Berger;Bioorg. Med Chem.,2009

3. Pharmacological comparative characterization of Rel-1017 (Esmethadone-Hcl) and other nmdar channel blockers in human heterodimeric N-Methyl-D-aspartate receptors;Bettini;Pharm. (Basel),2022

4. Trapping channel block of nmda-activated responses by amantadine and memantine;Blanpied;J. Neurophysiol.,1997

5. Protective effect of memantine on N-Methyl-D-aspartate receptor in dichlorvos-poisoned rat brain;Dai;Zhonghua Lao Dong Wei Sheng Zhi Ye Bing. Za Zhi,2004

同舟云学术

1.学者识别学者识别

2.学术分析学术分析

3.人才评估人才评估

"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370

www.globalauthorid.com

TOP

Copyright © 2019-2024 北京同舟云网络信息技术有限公司
京公网安备11010802033243号  京ICP备18003416号-3