Discovery of a highly potent, selective, orally bioavailable inhibitor of KAT6A/B histone acetyltransferases with efficacy against KAT6A-high ER+ breast cancer

Author:

Sharma Shikhar,Chung Chi-Yeh,Uryu Sean,Petrovic Jelena,Cao Joan,Rickard Amanda,Nady Nataliya,Greasley Samantha,Johnson Eric,Brodsky Oleg,Khan Showkhin,Wang Hui,Wang Zhenxiong,Zhang Yong,Tsaparikos Konstantinos,Chen Lei,Mazurek Anthony,Lapek John,Kung Pei-Pei,Sutton Scott,Richardson Paul F.,Greenwald Eric C.,Yamazaki Shinji,Jones Rhys,Maegley Karen A.,Bingham Patrick,Lam Hieu,Stupple Alexandra E.,Kamal Aileen,Chueh Anderly,Cuzzupe Anthony,Morrow Benjamin J.,Ren Bin,Carrasco-Pozo Catalina,Tan Chin Wee,Bhuva Dharmesh D.,Allan Elizabeth,Surgenor Elliot,Vaillant François,Pehlivanoglu Havva,Falk Hendrik,Whittle James R.,Newman Janet,Cursons Joseph,Doherty Judy P.,White Karen L.,MacPherson Laura,Devlin Mark,Dennis Matthew L.,Hattarki Meghan K.,De Silva Melanie,Camerino Michelle A.,Butler Miriam S.,Dolezal Olan,Pilling Patricia,Foitzik Richard,Stupple Paul A.,Lagiakos H. Rachel,Walker Scott R.,Hediyeh-Zadeh Soroor,Nuttall Stewart,Spall Sukhdeep K.,Charman Susan A.,Connor Theresa,Peat Thomas S.,Avery Vicky M.,Bozikis Ylva E.,Yang Yuqing,Zhang Ming,Monahan Brendon J.,Voss Anne K.,Thomas Tim,Street Ian P.,Dawson Sarah-Jane,Dawson Mark A.,Lindeman Geoffrey J.,Davis Melissa J.,Visvader Jane E.,Paul Thomas A.

Publisher

Elsevier BV

Subject

Clinical Biochemistry,Drug Discovery,Pharmacology,Molecular Biology,Molecular Medicine,Biochemistry

Reference109 articles.

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