A convenient method to synthesize phosphinic peptides containing an aspartyl or glutamyl aminophosphinic acid. Use of the phenyl group as the carboxyl synthon-Reference-Cited by-同舟云学术

A convenient method to synthesize phosphinic peptides containing an aspartyl or glutamyl aminophosphinic acid. Use of the phenyl group as the carboxyl synthon

Published:1999-12 Issue:51 Volume:55 Page:14635-14648
ISSN:0040-4020
Container-title:Tetrahedron
language:en
Short-container-title:Tetrahedron

Author:

Georgiadis Dimitris,Matziari Magdalini,Vassiliou Stamatia,Dive Vincent,Yiotakis Athanasios

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Reference32 articles.

1. Angiotensin-converting enzyme inhibitors. Mercaptan, carboxyalkyl dipeptide, and phosphinic acid inhibitors incorporating 4-substituted prolines

2. (Phosphinyloxy)acyl amino acid inhibitors of angiotensin converting enzyme (ACE). 1. Discovery of (S)-1-[6-amino-2-[[hydroxy(4-phenylbutyl)phosphinyl]oxy]-1-oxohexyl]-L-proline, a novel orally active inhibitor of ACE

3. Binding energetics of phosphorus-containing inhibitors of thermolysin

4. Phosphinic peptide analogues as potent inhibitors of Corynebacterium rathayii bacterial collagenase

5. Structure of astacin with a transition-state analogue inhibitor

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