In vitro and in vivo evaluation of polyoxyethylene indomethacin esters as dermal prodrugs

Author:

Bonina F.P.,Montenegro L.,De Caprariis P.,Palagiano F.,Trapani G.,Liso G.

Publisher

Elsevier BV

Subject

Pharmaceutical Science

Reference40 articles.

1. Prodrugs: Topical and Ocular Drug Delivery,1992

2. Percutaneous penetration enhancement: Physicochemical considerations and implications for prodrug design;Guy,1992

3. Transdermal delivery of levonorgestrel II: effect of prodrug structure on skin permeability in vitro;Friend;J. Control. Release,1988

4. Prodrugs for dermal delivery: solubility, molecular size, and functional group effects;Kasting,1992

5. Absorption of indomethacin and its calcium salt through rat skin: effect of penetration enhancers and relationship between in vivo and in vitro penetration;Ogiso;J. Pharmacobio-Dyn.,1986

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