TRPV1 antagonist with high analgesic efficacy: 2-Thio pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides-Reference-Cited by-同舟云学术

TRPV1 antagonist with high analgesic efficacy: 2-Thio pyridine C-region analogues of 2-(3-fluoro-4-methylsulfonylaminophenyl)propanamides

Published:2013-11 Issue:21 Volume:21 Page:6657-6664
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Ha Tae-Hwan,Ryu HyungChul,Kim Sung-Eun,Kim Ho Shin,Ann Jihyae,Tran Phuong-Thao,Hoang Van-Hai,Son Karam,Cui Minghua,Choi Sun,Blumberg Peter M.,Frank Robert,Bahrenberg Gregor,Schiene Klaus,Christoph Thomas,Frormann Sven,Lee Jeewoo

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference23 articles.

1. The Cloned Capsaicin Receptor Integrates Multiple Pain-Producing Stimuli

2. The capsaicin receptor: a heat-activated ion channel in the pain pathway

3. Vanilloid receptors on sensory nerves mediate the vasodilator action of anandamide

4. Direct activation of capsaicin receptors by products of lipoxygenases: Endogenous capsaicin-like substances

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