Bulleyaconitine A is a sensitive substrate and competitive inhibitor of CYP3A4: One of the possible explanations for clinical adverse reactions
Author:
Publisher
Elsevier BV
Subject
Pharmacology,Toxicology
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1. Development of a Novel CYP3A4 Classifier Model via Site of Metabolism (SOM)-based Molecular Docking, Multivariate Analysis and Molecular Dynamics of Known Substrates and Inhibitors;Journal of Computational Biophysics and Chemistry;2023-11-30
2. Clinical poisoning events involving yunaconitine may be highly correlated with metabolism-based interactions: A critical role of CYP3A4;Food and Chemical Toxicology;2023-09
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