Inhibition screening method of microsomal UGTs using the cocktail approach
Author:
Publisher
Elsevier BV
Subject
Pharmaceutical Science
Reference58 articles.
1. Role of human liver microsomes in in vitro metabolism of drugs – a review;Asha;Appl. Biochem. Biotechnol.,2010
2. Isolation and characterization of a novel cDNA encoding a human UDP-glucuronosyltransferase active on C-19 steroids;Beaulieu;J. Biol. Chem.,1996
3. The conduct of in vitro and in vivo drug–drug interaction studies: a pharmaceutical research and manufacturers of America (PhRMA) perspective;Bjornsson;Drug Metab. Dispos.,2003
4. The glucuronidation of Delta(4)-3-keto C19- and C21-hydroxysteroids by human liver microsomal and recombinant UDP-glucuronosyltransferases (UGTs): 6 alpha- and 21-hydroxyprogesterone are selective substrates for UGT2B7;Bowalgaha;Drug Metab. Dispos.,2007
5. Glucuronidation of nicotine and cotinine by UGT2B10: loss of function by the UGT2B10 codon 67 (Asp>Tyr) polymorphism;Chen;Cancer Res.,2007
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