Chapter 26 Mechanism-Based Inhibition of CYP3A4 and Other Cytochromes P450
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Elsevier
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2. Assessing and minimizing time-dependent inhibition of cytochrome P450 3A in drug discovery: A case study with melanocortin-4 receptor agonists
3. Contribution of Itraconazole Metabolites to Inhibition of CYP3A4 In Vivo
4. Qualitative Analysis of the Role of Metabolites in Inhibitory Drug−Drug Interactions: Literature Evaluation Based on the Metabolism and Transport Drug Interaction Database
5. Surface Plasmon Resonance Analysis of Antifungal Azoles Binding to CYP3A4 with Kinetic Resolution of Multiple Binding Orientations
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1. Computer-Aided (In Silico) Modeling of Cytochrome P450-Mediated Food–Drug Interactions (FDI);International Journal of Molecular Sciences;2022-07-31
2. Identification of chemical constituents of Zanthoxylum heitzii stem bark and their insecticidal activity against the malaria mosquito Anopheles gambiae;Parasites & Vectors;2015-10-01
3. CYP3A Time-Dependent Inhibition Risk Assessment Validated with 400 Reference Drugs;Drug Metabolism and Disposition;2011-03-07
4. Cobicistat (GS-9350): A Potent and Selective Inhibitor of Human CYP3A as a Novel Pharmacoenhancer;ACS Medicinal Chemistry Letters;2010-05-17
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