Practical application of 3-substituted-2,6-difluoropyridines in drug discovery: Facile synthesis of novel protein kinase C theta inhibitors-Reference-Cited by-同舟云学术

Practical application of 3-substituted-2,6-difluoropyridines in drug discovery: Facile synthesis of novel protein kinase C theta inhibitors

Published:2017-06 Issue:11 Volume:27 Page:2497-2501
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Katoh Taisuke,Tomata Yoshihide,Setoh Masaki,Sasaki Satoshi,Takai Takafumi,Yoshitomi Yayoi,Yukawa Tomoya,Nakagawa Hideyuki,Fukumoto Shoji,Tsukamoto Tetsuya,Nakada Yoshihisa

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference34 articles.

1. New heterocyclic analogues of 4-(2-chloro-5-methoxyanilino)quinazolines as potent and selective c-Src kinase inhibitors

2. Novel pyridinyl and pyrimidinylcarbazole sulfonamides as antiproliferative agents

3. First synthesis of 1-deazacytidine, the C-nucleoside analogue of cytidine

4. The Reactivity of 2-Fluoro- and 2-Chloropyridines toward Sodium Ethoxide: Factors Governing the Rates of Nucleophilic (Het)Aromatic Substitutions

5. An efficient access to 3,6-disubstituted 1H-pyrazolo[3,4-b]pyridines via a one-pot double SNAr reaction and pyrazole formation

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5. Facile Preparation of 3-Substituted-2,6-difluoropyridines and Application to the Synthesis of 2,3,6-Trisubstituted Pyridines for PKCθ Inhibitors;Journal of Synthetic Organic Chemistry, Japan;2020-02-01