Conformationally constrained farnesoid X receptor (FXR) agonists: Naphthoic acid-based analogs of GW 4064-Reference-Cited by-同舟云学术

Conformationally constrained farnesoid X receptor (FXR) agonists: Naphthoic acid-based analogs of GW 4064

Published:2008-08 Issue:15 Volume:18 Page:4339-4343
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Akwabi-Ameyaw Adwoa,Bass Jonathan Y.,Caldwell Richard D.,Caravella Justin A.,Chen Lihong,Creech Katrina L.,Deaton David N.,Jones Stacey A.,Kaldor Istvan,Liu Yaping,Madauss Kevin P.,Marr Harry B.,McFadyen Robert B.,Miller Aaron B.,III Frank Navas,Parks Derek J.,Spearing Paul K.,Todd Dan,Williams Shawn P.,Wisely G. Bruce

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference39 articles.

1. FXR signaling in metabolic disease

2. Identification of a Nuclear Receptor for Bile Acids

3. Bile Acids: Natural Ligands for an Orphan Nuclear Receptor

4. Identification of a nuclear receptor that is activated by farnesol metabolites

5. Immunolocalization of farnesoid X receptor (FXR) in mouse tissues using tissue microarray

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