Identification of novel benzimidazole derivatives as highly potent AMPK activators with anti-diabetic profiles

Author:

Tamura Yuusuke,Morita Ippei,Hinata Yu,Kojima Eiichi,Sasaki Yoshikazu,Wada Toshihiro,Asano Mutsumi,Fujioka Masahiko,Hayasaki-Kajiwara Yoko,Iwasaki Takanori,Matsumura Kenichi

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference15 articles.

1. World Health Organization, Fact sheets, Diabetes, 10 November 2021, retrieved from https://www.who.int/news-room/fact-sheets/detail/diabetes.

2. AMPK in Health and Disease;Steinberg;Physiol Rev,2009

3. Exercise, GLUT4, and skeletal muscle glucose uptake;Richter;Physiol Rev,2013

4. Pharmacological AMPK activation induces transcriptional responses congruent to exercise in skeletal and cardiac muscle, adipose tissues and liver;Muise;PLoS One,2019

5. Role of Skeletal Muscle in Insulin Resistance and Glucose Uptake;Merz;Compr Physiol.,2020

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