PD 165929 — the first high affinity non-peptide neuromedin-B (NMB) receptor selective antagonist-Reference-Cited by-同舟云学术

PD 165929 — the first high affinity non-peptide neuromedin-B (NMB) receptor selective antagonist

Published:1996-11 Issue:21 Volume:6 Page:2617-2622
ISSN:0960-894X
Container-title:Bioorganic & Medicinal Chemistry Letters
language:en
Short-container-title:Bioorganic & Medicinal Chemistry Letters

Author:

Eden J.M.,Hall M.D.,Higginbottom M.,Horwell D.C.,Howson W.,Hughes J.,Jordan R.E.,Lewthwaite R.A.,Martin K.,McKnight A.T.,O'Toole J.C.,Pinnock R.D.,Pritchard M.C.,Suman-Chauhan N.,Williams S.C.

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference19 articles.

1. The asymmetric synthesis of non-peptide CCK-A receptor agonists

2. Rationally designed "dipeptoid" analogs of CCK. .alpha.-Methyltryptophan derivatives as highly selective and orally active gastrin and CCK-B antagonists with potent anxiolytic properties

3. The development of a novel series of non-peptide tachykinin NK3 receptor selective antagonists

4. The ‘peptoid’ approach to the design of non-peptide, small molecule agonists and antagonists of neuropeptides

5. Rational design of high affinity tachykinin NK2 receptor antagonists

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