Novel 2-arylbenzothiazole DNA gyrase inhibitors: Synthesis, antimicrobial evaluation, QSAR and molecular docking studies
Author:
Funder
National Research Centre
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry
Reference42 articles.
1. New N-phenylpyrrolamide DNA gyrase B inhibitors: optimization of efficacy and antibacterial activity;Durcik;Eur. J. Med. Chem.,2018
2. Pyridine-3-carboxamide-6-yl-ureas as novel inhibitors of bacterial DNA gyrase: structure based design, synthesis, SAR and antimicrobial activity;Yule;Eur. J. Med. Chem.,2014
3. Epidemiological and resistance issues in multidrug-resistant staphylococci and enterococci;Leclercq;Clin. Microbiol. Infect.,2009
4. Discovery of benzothiazole scaffold-based DNA gyrase B inhibitors;Gjorgjieva;J. Med. Chem.,2016
5. Design, synthesis and biological evaluation of alpha-substituted isonipecotic acid benzothiazole analogues as potent bacterial type II topoisomerase inhibitors;Axford;Bioorg. Med. Chem. Lett.,2013
Cited by 19 articles. 订阅此论文施引文献 订阅此论文施引文献,注册后可以免费订阅5篇论文的施引文献,订阅后可以查看论文全部施引文献
1. Schematic-portfolio of potent anti-microbial scaffolds targeting DNA gyrase: Unlocking ways to overcome resistance;International Journal of Biological Macromolecules;2024-01
2. Design, docking, molecular dynamics, synthesis and antimicrobial studies on quinoline derivatives and some isosteres;Journal of Molecular Structure;2023-12
3. The influence of proton-donor solvent on [4+2] benzannulation reaction of dienal with tertiary enaminone;Computational and Theoretical Chemistry;2023-11
4. Recent insights into antibacterial potential of benzothiazole derivatives;Medicinal Chemistry Research;2023-05-29
5. Strategies towards the Synthesis of 2‐Ketoaryl Azole Derivatives using C‐H Functionalization Approach and 1,2‐Bis‐Nucleophile Precursors;Asian Journal of Organic Chemistry;2023-03-24
1.学者识别学者识别
2.学术分析学术分析
3.人才评估人才评估
"同舟云学术"是以全球学者为主线,采集、加工和组织学术论文而形成的新型学术文献查询和分析系统,可以对全球学者进行文献检索和人才价值评估。用户可以通过关注某些学科领域的顶尖人物而持续追踪该领域的学科进展和研究前沿。经过近期的数据扩容,当前同舟云学术共收录了国内外主流学术期刊6万余种,收集的期刊论文及会议论文总量共计约1.5亿篇,并以每天添加12000余篇中外论文的速度递增。我们也可以为用户提供个性化、定制化的学者数据。欢迎来电咨询!咨询电话:010-8811{复制后删除}0370
www.globalauthorid.com
TOP
Copyright © 2019-2024 北京同舟云网络信息技术有限公司 京公网安备11010802033243号 京ICP备18003416号-3