Design, synthesis and bioactivity evaluation of selenium-containing PI3Kδ inhibitors

Author:

Gao Li,Chuai Hongyan,Ma Mengyan,Zhang San-Qi,Zhang Jiye,Li Jiyu,Wang Yang,Xin Minhang

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference42 articles.

1. PI3K in cancer: divergent roles of isoforms, modes of activation and therapeutic targeting;Thorpe;Nat. Rev. Cancer,2015

2. Synergy in activating class I PI3Ks;Burke;Trends Biochem. Sci.,2015

3. Targeting the phosphoinositide 3 kinase pathway in cancer;Liu;Nat. Rev. Drug Discov.,2010

4. Class I phosphatidylinositol-3-kinase inhibitors for cancer therapy;Zhao;Acta Pharm. Sin. B,2017

5. 6-Aryl substituted 4-(4-cyanomethyl) phenylamino quinazolines as a new class of isoform-selective PI3K-alpha inhibitors;Yadav;Eur. J. Med. Chem.,2016

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