A novel class of pyrazole analogues as aurora kinase A inhibitor: design, synthesis, and anticancer evaluation

Author:

Yevale Digambar B.,Teraiya Nishith,Lalwani Twinkle D.,Ameta Rakesh Kumar,Sangani Chetan B.

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Molecular Biology,Biochemistry

Reference39 articles.

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3. 3-Cyano-6-(5-methyl-3-pyrazoloamino)pyridines: Selective Aurora A kinase inhibitors;Ando;Bioorg. Med. Chem. Lett.,2010

4. Discovery of a potent, selective, and orally bioavailable pyridinyl-pyrimidine phthalazine aurora kinase inhibitor;Cee;J. Med. Chem.,2010

5. Specific small-molecule activator of Aurora kinase A induces autophosphorylation in a cell-free system;Kishore;J. Med. Chem.,2008

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