Inhibiting 5-Fluorouracil Breakdown: A Broken Down Approach to 5-Fluorouracil Modulation

Author:

Schilsky Richard L.

Publisher

Elsevier BV

Subject

Gastroenterology,Oncology

Reference16 articles.

1. Response to fluorouracil therapy in cancer patients: the role of tumoral dihydropyrimidine dehydrogenase activity;Etienne;J Clin Oncol,1995

2. 5-Ethynyluracil (776C85): inactivation of dihydropyrimidine dehydrogenase in vivo;Spector;Biochem Pharmacol,1993

3. Mechanism- based inactivation of dihydropyrimidine dehydrogenase by 5-ethynyluracil;Porter;J Biol Chem,1992

4. 5-Ethynyluracil (776C85): a potent modulator of the pharmacokinetics and antitumor efficacy of 5-fluorouracil;Baccanari;Proc Natl Acad Sci U S A,1993

5. 5-Ethynyluracil (776C85): modulation of 5-fluorouracil efficacy and therapeutic index in rats bearing advanced colorectal carcinoma;Cao;Cancer Res,1994

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