Synthesis and characterization of the two enantiomers of a chiral sigma-1 receptor radioligand: (S)-(+)- and (R)-(-)-[18F]FBFP-Reference-Cited by-同舟云学术

Synthesis and characterization of the two enantiomers of a chiral sigma-1 receptor radioligand: (S)-(+)- and (R)-(-)-[18F]FBFP

Published:2022-07 Issue:7 Volume:33 Page:3543-3548
ISSN:1001-8417
Container-title:Chinese Chemical Letters
language:en
Short-container-title:Chinese Chemical Letters

Author:

Wang Tao^ORCID,Zhang Ying,Zhang Xiaojun,Chen Leyuan,Zheng Mingqiang,Zhang Jinming,Brust Peter^ORCID,Deuther-Conrad Winnie,Huang Yiyun,Jia Hongmei^ORCID

Funder

National Natural Science Foundation of China

Natural Science Foundation of Beijing Municipality

Publisher

Elsevier BV

Subject

General Chemistry

Reference49 articles.

1. Cloning and Functional Expression of the Human Type 1 Sigma Receptor (hSigmaR1)

2. Purification, molecular cloning, and expression of the mammalian sigma1-binding site.

3. Crystal structure of the human σ1 receptor

4. Sigma-1 Receptor Chaperones at the ER- Mitochondrion Interface Regulate Ca2+ Signaling and Cell Survival

5. Structural basis for σ1 receptor ligand recognition

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