Design, synthesis and biological evaluation of tricyclic pyrazolo[1,5-c][1,3]benzoxazin-5(5H)-one scaffolds as selective BuChE inhibitors
Author:
Affiliation:
1. School of Pharmacy, Anhui Medical University, Hefei, PR China;
2. Lujiang County People's Hospital, Lujiang, Anhui, PR China;
3. Anhui Prevention and Treatment Center for Occupational Disease, Hefei, PR China
Funder
Anhui University Natural Science Research Project
Publisher
Informa UK Limited
Subject
Drug Discovery,Pharmacology,General Medicine
Link
https://www.tandfonline.com/doi/pdf/10.1080/14756366.2018.1488696
Reference45 articles.
1. Alzheimer's disease
2. Cortical pyroglutamate amyloid-β levels and cognitive decline in Alzheimer's disease
3. 2016 Alzheimer's disease facts and figures
4. Biochemistry of Amyloid -Protein and Amyloid Deposits in Alzheimer Disease
5. Tau phosphorylation and aggregation in Alzheimer's disease pathology
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