New potent steroid sulphatase inhibitors based on 6-(1-phenyl-1H-1,2,3-triazol-4-yl)naphthalen-2-yl sulphamate derivatives

Author:

Ciupak Olga1,Daśko Mateusz2ORCID,Biernacki Karol1ORCID,Rachon Janusz1ORCID,Masłyk Maciej3,Kubiński Konrad3ORCID,Martyna Aleksandra3ORCID,Demkowicz Sebastian1ORCID

Affiliation:

1. Department of Organic Chemistry, Faculty of Chemistry, Gdańsk University of Technology, Gdańsk, Poland

2. Department of Inorganic Chemistry, Faculty of Chemistry, Gdańsk University of Technology, Gdańsk, Poland

3. Department of Molecular Biology, The John Paul II Catholic University of Lublin, Lublin, Poland

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Reference37 articles.

1. IARC: CANCER FACT SHEETS [Internet]. Lyon (France): International Agency for Research on Cancer. Available from: https://gco.iarc.fr/today/factsheets-cancers [last accessed 10 May 2020].

2. NCI [Internet]. Maryland (U.S.): National Cancer Institiute. Available from: https://seer.cancer.gov/statfacts/html/breast.html [last accessed on 10 May 2020].

3. Steroid sulfatase: A pivotal player in estrogen synthesis and metabolism

4. Sulfatase inhibitors for recidivist breast cancer treatment: A chemical review

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