Design, synthesis, molecular modeling, and biological evaluations of novel chalcone based 4-Nitroacetophenone derivatives as potent anticancer agents targeting EGFR-TKD

Author:

Mir Showkat Ahmad1,Murmu Narayan2,Meher Rajesh Kumar1,Baitharu Iswar3,Nayak Binata1,Khan Andleeb4,Khan Mohammad Imran56,Abdulaal Wesam H.78

Affiliation:

1. School of Life Sciences, Sambalpur University, Sambalpur, India

2. School of Chemistry, Sambalpur University, Sambalpur, India

3. Department of Environmental Sciences, Sambalpur University, Sambalpur, India

4. Department of Biosciences, Faculty of Science, Integral University, Lucknow, India

5. Department of Biochemistry, Faculty of Science, King Abdulaziz University, Jeddah, Saudi Arabia

6. Centre for Artificial Intelligence in Precision Medicines, King Abdulaziz University, Jeddah, Saudi Arabia

7. Department of Biochemistry, Faculty of Science, Cancer and Mutagenesis Unit, King Fahd Medical Research Center, King Abdulaziz University, Jeddah, Saudi Arabia

8. Center of Excellence for Drug Research and Pharmaceutical Industries, King Abdulaziz University, Jeddah, Saudi Arabia

Funder

Institutional Fund Projects

Ministry of Education and King Abdulaziz University

Publisher

Informa UK Limited

Subject

Molecular Biology,General Medicine,Structural Biology

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