The in vitro pharmacological profile of TD-1211, a neutral opioid receptor antagonist-Reference-Cited by-同舟云学术

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The in vitro pharmacological profile of TD-1211, a neutral opioid receptor antagonist

Published:2013-04-04 Issue:6 Volume:386 Page:479-491
ISSN:0028-1298
Container-title:Naunyn-Schmiedeberg's Archives of Pharmacology
language:en
Short-container-title:Naunyn-Schmiedeberg's Arch Pharmacol

Author:

Tsuruda Pamela R.,Vickery Ross G.,Long Daniel D.,Armstrong Scott R.,Beattie David T.

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology,General Medicine

Link

http://link.springer.com/content/pdf/10.1007/s00210-013-0850-7.pdf

Reference54 articles.

1. Armstrong SR, Campbell CB, Richardson CL, Vickery RG, Tsuruda PR, Long DD, Hegde SS, Beattie DT (2013) The in vivo pharmacology of TD-1211, a peripherally-selective opioid receptor antagonist in development for the treatment of opioid-induced constipation. Naunyn-Schmiedeberg’s Arch Pharm. doi: 10.1007/s00210-013-0844-5

2. Arunlakshana O, Schild HO (1959) Some quantitative uses of drug antagonists. Br J Pharmacol Chemotherap 14:48–58

3. Beattie DT, Cheruvu M, Mai N, O’Keefe M, Johnson-Rabidoux S, Peterson C, Kaufman E, Vickery R (2007) The in vitro pharmacology of the peripherally restricted opioid receptor antagonists, alvimopan, ADL 08–0011 and methylnaltrexone. Naunyn Schmiedeberg’s Arch Pharmacol 375:205–220

4. Brent PJ, Chahl LA, Cantarella PA, Kavanagh C (1993) The kappa-opioid receptor agonist U50,488H induces acute physical dependence in guinea-pigs. Eur J Pharmacol 241:149–156

5. Brock C, Olesen SS, Olesen AE, Frokjaer JB, Andresen T, Drewes AM (2012) Opioid-induced bowel dysfunction. Drugs 72:1847–1865

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