Synthesis, anticancer evaluation and docking studies of novel adamantanyl-1,3,4-oxadiazol hybrid compounds as Aurora-A kinase inhibitors
Author:
Publisher
Springer Science and Business Media LLC
Subject
Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics
Link
https://link.springer.com/content/pdf/10.1007/s00044-023-03145-4.pdf
Reference44 articles.
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2. Pradhan T, Gupta O, Singh G, Monga V. Aurora kinase inhibitors as potential anticancer agents: recent advances. Eur J Med Chem. 2021;221:113495. https://doi.org/10.1016/j.ejmech.2021.113495.
3. Carry J-C, Clerc F, Minoux H, Schio L, Mauger J, Nair A, et al. SAR156497, an exquisitely selective inhibitor of aurora kinases. J Med Chem. 2015;58:362–75. https://doi.org/10.1021/jm501326k.
4. Chi Y-H, Yeh TK, Ke YY, Lin WH, Tsai CH, Wang WP, et al. Discovery and synthesis of a pyrimidine-based Aurora kinase inhibitor to reduce levels of MYC Oncoproteins. J Med Chem. 2021;64:7312–30. https://doi.org/10.1021/acs.jmedchem.0c01806.
5. Islam MS, Wang C, Zheng J, Paudyal N, Zhu Y, Sun H. The potential role of tubeimosides in cancer prevention and treatment. Eur J Med Chem. 2019;162:109–21. https://doi.org/10.1016/j.ejmech.2018.11.001.
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