Metabolic profile of XK469 (2(R)-[4-(7-chloro-2-quinoxalinyl)oxyphenoxy]-propionic acid; NSC698215) in patients and in vitro: low potential for active or toxic metabolites or for drug–drug interactions

Author:

Anderson Lawrence W.,Collins Jerry M.,Klecker Raymond W.,Katki Aspandiar G.,Parchment Ralph E.,Boinpally Ramesh R.,LoRusso Patricia M.,Ivy S. Percy

Publisher

Springer Science and Business Media LLC

Subject

Pharmacology (medical),Cancer Research,Pharmacology,Toxicology,Oncology

Reference24 articles.

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2. Beedham C, Miceli JJ, Obach RS (2003) Ziprasidone metabolism, aldehyde oxidase, and clinical implications. J Psychopharmacol 23:229–232

3. Chabner BA (2001) Cytidine analogues. In: Chabner BA, Longo DL (eds) Cancer chemotherapy and biotherapy. Lippincott Williams & Wilkins, Philadelphia, pp 213–233

4. Collins JM (2000) Cytochrome P-450 and other determinants of pharmacokinetics, toxicity, and efficacy in humans. Clin Cancer Res 6:1203–1204

5. Collins JM (2000) Prediction of drug interactions from in vitro studies: regulatory viewpoint. In: Levy RH, Thummel KE, Trager WF, Hansten P, Eichelbaum M (eds) Metabolic drug interactions. Lippincott-Raven, Philadelphia, pp 41–47

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