Assay of GTPγS Binding in Autoradiography

Author:

Gabaglio Marina,Prini Pamela,Zamberletti Erica,Rubino Tiziana,Parolaro Daniela

Publisher

Springer US

Reference10 articles.

1. Vasavda C, Zaccor NW, Scherer PC, Sumner CJ, Snyder SH (2017) Measuring G-protein-coupled receptor signaling via radio-labeled GTP binding. J Vis Exp 124:55561

2. Yang D, Zhou Q, Labroska V et al (2021) G protein-coupled receptors: structure- and function-based drug discovery. Sig Transduct Target Ther 6:7

3. Sriram K, Insel PA (2018) G protein-coupled receptors as targets for approved drugs: how many targets and how many drugs? Mol Pharmacol 93:251–258

4. Sóvágó J, Dupuis DS, Gulyás B et al (2001) An overview on functional receptor autoradiography using 35[ S]GTPgS. Brain Res Brain Res Rev 38:149–164

5. Zarbin MA, Palacios JM, Wamsley JK et al (1983) Axonal transport of b-adrenergic receptors. Antero- and retrogradely transported receptors differ in agonist affinity and nucleotide sensitivity. Mol Pharmacol 24:341–348

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